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HS 024

CAT: 0013-GTR19157590-01Size: 200 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19157590-01Size:200 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively) . Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.
CAS Number
212370-59-7
Purity
>98% (HPLC)
Solubility
Water:0.50 mg/mL
Smiles
CCCC[C@@H]1NC (=O) [C@H] (CSSC[C@H] (NC (=O) CNC (=O) [C@H] (Cc2c[nH]c3ccccc23) NC (=O) [C@H] (CCCNC (N) =N) NC (=O) [C@@H] (Cc2ccc3ccccc3c2) NC (=O) [C@H] (Cc2c[nH]cn2) NC (=O) [C@H] (CCCNC (N) =N) NC1=O) C (N) =O) NC (C) =O
Molecular Formula
C58H79N19O10S2
Molecular Weight
1266.5
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.

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