GPR41 modulator 1
CAT:
804-HY-163530
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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GPR41 modulator 1
- CAS Number: 3050768-93-6
- UNSPSC Description: GPR41 modulator 1 (compound 10ak) is a potent GPR41 modulator with an EC50 value of 0.679 µM. GPR41 modulator 1 shows agonistic modulator activity[1].
- Target Antigen: Free Fatty Acid Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein
- Applications: Metabolism-protein/nucleotide metabolism
- Field of Research: Metabolic Disease; Inflammation/Immunology
- Assay Protocol: https://www.medchemexpress.com/gpr41-modulator-1.html
- Smiles: FC1=CC(F)=CC(C2=CC=C(O2)C3C(C(NC4=C(C=CC=C4)C)=O)=C(NC5=C3C(CCC5)=O)C)=C1
- Molecular Weight: 474.50
- References & Citations: [1]Inuki S, et al. Structure-activity relationship studies of tetrahydroquinolone derivatives as GPR41 modulators. Bioorg Med Chem Lett. 2024 Jul 15;107:129758.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported