IK-930

• Description:

  IK-930 (compound I-32) is a potent and orally active TEAD inhibitor with an EC50 value of [1].

• UNSPSC:

  12352005

• Target:

  YAP

• Type:

  Reference compound

• Related Pathways:

  Stem Cell/Wnt

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/ik-930.html

• Purity:

  99.39

• Solubility:

  DMSO : 100 mg/mL (ultrasonic)

• Smiles:

  O=S(NC)(C1=CC(C2=CN(C)C=N2)=C(NCC3=CC=C(C(F)(F)F)C=C3)C=C1)=O

• Molecular Formula:

  C19H19F3N4O2S

• Molecular Weight:

  424.44

• References & Citations:

  [1]Alfredo C. Castro, et al. Tead inhibitors and uses thereof. WO2020243415A2.

• Shipping Conditions:

  Room Temperature

• Storage Conditions:

  -20°C, 3 years; 4°C, 2 years (Powder)

• Scientific Category:

  Reference compound1

• Clinical Information:

  Phase 1

• CAS Number:

  2563892-44-2