CAC 253 acetate

• Target:

  Amylin Receptor

• Related Pathways:

  GPCR/G Protein

• Purity:

  0.9999

• Bioactivity:

  CAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.

• Smiles:

  C[C@@H](O)[C@H]1C(N[C@@H](CC2=CC=C(O)C=C2)C(N3CCC[C@H]3C(N[C@@H](CCCNC(N)=N)C(N[C@@H]([C@H](O)C)C(N[C@@H](CC(N)=O)C(N[C@@H]([C@H](O)C)C(NCC(N[C@@H](CO)C(N[C@@H](CC(N)=O)C(N[C@@H]([C@H](O)C)C(N[C@@H](CC4=CC=C(O)C=C4)C(N[C@H](C(N)=O)CSSC[C@H](N)C(N[C@@H](CC(C)C)C(NCC(N[C@@H](CCCNC(N)=N)C(N[C@@H](CC(C)C)C(N[C@@H](CO)C(N[C@@H](CCC(N)=O)C(N[C@@H](CCC(O)=O)C(N[C@@H](CC(C)C)C(N[C@@H](CC5=CNC=N5)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CC(C)C)C(N[C@@H](CCC(N)=O)C(N1)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O.CC(O)=O

• Molecular Formula:

  C128H206N42O42S2

• Molecular Weight:

  3069.39

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C