[Ala17]-MCH

• Target:

  GPCR|||Melanin-concentrating Hormone Receptor (MCHR)

• Related Pathways:

  Endocrinology/Hormones|||GPCR/G Protein

• Bioactivity:

  Potent melanin-concentrating hormone (MCH) receptor agonist (EC50 values are 17 and 54 nM at MCH1 and MCH2 receptors respectively) . Displays some selectivity towards MCH1 over MCH2 (Ki values are 0.16 and 34 nM respectively) .

• Smiles:

  O=C1N2C (C (=O) N[C@H] (C (N[C@H] (C (N[C@H] (C (N[C@@H] ([C@H] (C) C) C (O) =O) =O) CCC (N) =O) =O) C) =O) CSSC[C@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@H] (CC3=CC=CC=C3) NC ([C@H] (CC (O) =O) N) =O) =O) CC (O) =O) =O) CCSC) =O) CC (C) C) =O) CCCNC (=N) N) =O) C (=O) N[C@@H] (CCSC) C (=O) N[C@@H] (CC (C) C) C (=O) NCC (=O) N[C@@H] (CCCNC (=N) N) C (=O) N[C@@H] ([C@@H] (C) C) C (=O) N[C@@H] (CC4=CC=C (O) C=C4) C (=O) N[C@H]1CCCNC (=N) N) (CCC2) [H]

• Molecular Formula:

  C97H155N29O26S4

• Molecular Weight:

  2271.71

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  359784-84-2