Products for Research Use Only

MCH (human, mouse, rat) TFA

CAT: 0931-T75846-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T75846-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
GPCR, Melanin-concentrating Hormone Receptor (MCHR)
Related Pathways
Endocrinology/Hormones, GPCR/G Protein
Bioactivity
MCH (human, mouse, rat) TFA is a potent peptide agonist for MCH receptors, exhibiting binding IC50 values of 0.3 nM for MCH1R and 1.5 nM for MCH2R. It is particularly effective against MCH-2R in a CHO cell line, with functional activation EC50 values of 3.9 nM for MCH-1R and 0.1 nM for MCH-2R, as evidenced by intracellular calcium mobilization measured with FLIPR [1].
Molecular Formula
C107H161F3N30O28S4
Molecular Weight
2500.86
Shipping Conditions
Ice Packs
Storage Temperature
-20°C