TC-MCH 7c

• Target:

  Melanin-concentrating Hormone Receptor (MCHR) |||GPCR

• Related Pathways:

  Endocrinology/Hormones|||GPCR/G Protein

• Purity:

  0.9954

• Bioactivity:

  TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance of 5.6 nM against hMCH1R, and TC-MCH 7c is a phenylpyridone derivative with MCH1R Ki of 3.4 nM against human. In mice, MCH1R Ki was 3.0 nM.

• Smiles:

  Fc1ccc(COc2ccn(-c3ccc(OCCN4CCCC4)cc3)c(=O)c2)cc1

• Molecular Formula:

  C24H25FN2O3

• Molecular Weight:

  408.47

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  864756-35-4