[Ala17]-MCH TFA

• Target:

  GPCR|||Melanin-concentrating Hormone Receptor (MCHR)

• Related Pathways:

  Endocrinology/Hormones|||GPCR/G Protein

• Bioactivity:

  [Ala17]-MCH TFA, a selective ligand for MCHR 1 (K i =0.16 nM) over MCHR 2 (K i =34 nM), is an analogue of MCH. When labeled with a [Eu 3+ chelate], [Ala17]-MCH exhibits high affinity for MCHR 1 (K d =0.37 nM) and negligible binding affinity for MCHR 2.

• Molecular Formula:

  C99H156F3N29O28S4

• Molecular Weight:

  2385.73

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C