PCLX-001

• Target:

  Others

• Related Pathways:

  Others

• Purity:

  0.996

• Bioactivity:

  PCLX-001 is a small-molecule compound that acts as an orally active inhibitor of N-myristoyltransferase (NMT), specifically targeting NMT1 and NMT2 with IC50 values of 5 nM and 8 nM, respectively. This compound demonstrates anti-tumor effects and effectively inhibits the early signaling of B-cell receptor (BCR) . Consequently, PCLX-001 is a valuable tool for researching B-cell malignancies [1] [2].

• Smiles:

  N(S(=O)(=O)C1=C(Cl)C=C(C=C1Cl)C=2C=C(N=CC2)N3CCNCC3)C=4C(CC(C)C)=NN(C)C4C

• Molecular Formula:

  C24H30Cl2N6O2S

• Molecular Weight:

  537.51

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1215011-08-7