RLX-33

• Target :

  RXFP receptor|||ERK

• Related Pathways :

  MAPK|||GPCR/G Protein

• Purity :

  0.9989

• Bioactivity :

  RLX-33 is a potent and selective antagonist of relaxin family peptide 3 (RXFP3) that crosses the blood-brain barrier and also blocks relaxin 3-induced ERK1/2 phosphorylation. RLX-33 can block the increase in food intake induced by the RXFP3 selective agonist R3/I5 in rats.RLX-33 can be used to study the metabolic syndrome.

• Smiles :

  N(C(=O)C1CN(CC2=CC=CO2)C(=O)C1)C3=CC=C(C4=NC(=NO4)C5=CC=C(Cl)C=C5)C=C3

• Molecular Formula :

  C24H19ClN4O4

• Molecular Weight :

  462.89

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2784577-71-3