RLX-33

• Target:

  RXFP receptor|||ERK

• Related Pathways:

  MAPK|||GPCR/G Protein

• Purity:

  0.9989

• Bioactivity:

  RLX-33 is a potent and selective antagonist of relaxin family peptide 3 (RXFP3) that crosses the blood-brain barrier and also blocks relaxin 3-induced ERK1/2 phosphorylation. RLX-33 can block the increase in food intake induced by the RXFP3 selective agonist R3/I5 in rats.RLX-33 can be used to study the metabolic syndrome.

• Smiles:

  N (C (=O) C1CN (CC2=CC=CO2) C (=O) C1) C3=CC=C (C4=NC (=NO4) C5=CC=C (Cl) C=C5) C=C3

• Molecular Formula:

  C24H19ClN4O4

• Molecular Weight:

  462.89

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2784577-71-3