PKM2 activator 3

• Target:

  Others|||PKM

• Related Pathways:

  Others|||Metabolism

• Bioactivity:

  PKM2 activator 3 is a highly potent compound that activates PKM2, with an AC 50 value of 90 nM. It exhibits excellent Caco-2 permeability, a low efflux ratio, and remarkable microsomal stability. PKM2 activator 3 is particularly valuable for anticancer research purposes [1]. (AC 50: the concentration at which 50% enzyme activation occurs.)

• Smiles:

  FC=1C=C2C (=CC1S (NC3=CC (Cl) =C (F) C=C3) (=O) =O) CCC (=O) N2

• Molecular Formula:

  C15H11ClF2N2O3S

• Molecular Weight:

  372.77

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1346113-84-5