Products for Research Use Only

PKM2 activator 3

CAT: 0931-T61504-01Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T61504-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1346113-84-5
Target
Others, PKM
Related Pathways
Others, Metabolism
Bioactivity
PKM2 activator 3 is a highly potent compound that activates PKM2, with an AC 50 value of 90 nM. It exhibits excellent Caco-2 permeability, a low efflux ratio, and remarkable microsomal stability. PKM2 activator 3 is particularly valuable for anticancer research purposes [1]. (AC 50: the concentration at which 50% enzyme activation occurs.)
Smiles
FC=1C=C2C(=CC1S(NC3=CC(Cl)=C(F)C=C3)(=O)=O)CCC(=O)N2
Molecular Formula
C15H11ClF2N2O3S
Molecular Weight
372.77
Shipping Conditions
Ice Packs
Storage Temperature
-20°C