PKM2 activator 3

• CAS Number :

  1346113-84-5

• Target :

  Others|||PKM

• Related Pathways :

  Others|||Metabolism

• Bioactivity :

  PKM2 activator 3 is a highly potent compound that activates PKM2, with an AC 50 value of 90 nM. It exhibits excellent Caco-2 permeability, a low efflux ratio, and remarkable microsomal stability. PKM2 activator 3 is particularly valuable for anticancer research purposes [1]. (AC 50: the concentration at which 50% enzyme activation occurs.)

• Smiles :

  FC=1C=C2C(=CC1S(NC3=CC(Cl)=C(F)C=C3)(=O)=O)CCC(=O)N2

• Molecular Formula :

  C15H11ClF2N2O3S

• Molecular Weight :

  372.77

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C