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ARV-771

CAT: 0931-T5435-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T5435-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1949837-12-0
Target
Epigenetic Reader Domain, PROTACs
Related Pathways
PROTAC, Chromatin/Epigenetic
Purity
0.9969
Bioactivity
ARV-771 is an effective BET degrader based on PROTAC technology. The Kd for BRD2 (1), BRD2 (2), BRD3 (1), BRD3 (2), BRD4 (1) and BRD4 (2) are 34 and 4.7 respectively. , 8.3, 7.6, 9.6 and 7.6 nM.
Smiles
CC=1C2=C(N3C([C@H](CC(NCCOCCCOCC(N[C@H](C(=O)N4[C@H](C(N[C@@H](C)C5=CC=C(C=C5)C=6SC=NC6C)=O)C[C@@H](O)C4)C(C)(C)C)=O)=O)N=C2C7=CC=C(Cl)C=C7)=NN=C3C)SC1C
Molecular Formula
C49H60ClN9O7S2
Molecular Weight
986.64
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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