GNE-375

• Target:

  Epigenetic Reader Domain|||Carboxypeptidase|||CDK

• Related Pathways:

  Proteases/Proteasome|||Chromatin/Epigenetic|||Cell Cycle/Checkpoint

• Purity:

  0.9932

• Bioactivity:

  GNE-375 is a selective and potent BRD9 inhibitor (IC50: 5 nM) .GNE-375 inhibits BRD4, TAF1, and CECR2, and can be used to study epigenetic resistance.

• Smiles:

  COc1cc (c (OC) cc1C (=O) N1CCOCC1) -c1cn (C\C=C\C) c (=O) c2[nH]c (C) cc12

• Molecular Formula:

  C25H29N3O5

• Molecular Weight:

  451.51

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1926989-06-1