GNE-375
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


GNE-375
CAS Number :
1926989-06-1Target :
Epigenetic Reader Domain|||Carboxypeptidase|||CDKRelated Pathways :
Proteases/Proteasome|||Chromatin/Epigenetic|||Cell Cycle/CheckpointPurity :
0.9932Bioactivity :
GNE-375 is a selective and potent BRD9 inhibitor (IC50: 5 nM) .GNE-375 inhibits BRD4, TAF1, and CECR2, and can be used to study epigenetic resistance.Smiles :
COc1cc(c(OC)cc1C(=O)N1CCOCC1)-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12Molecular Formula :
C25H29N3O5Molecular Weight :
451.51Shipping Conditions :
Cool packStorage Temperature :
-20°C

