Products for Research Use Only

GNE-616

CAT: 0931-T11439-01Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T11439-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
2349371-81-7
Target
Sodium Channel, Others
Related Pathways
Membrane transporter/Ion channel, Others
Bioactivity
GNE-616 is a highly potent, metabolically stable, orally bioavailable, and subtype-selective Nav1.7 inhibitor [Ki: 0.79 nM, Kd: 0.38 nM for hNav1.7] for the treatment of chronic pain.
Smiles
C(F)(F)(F)[C@@H]1C[C@@H](N(CC1)[C@@H]2C=3C(=CC(S(NC=4C=CN=CN4)(=O)=O)=C(F)C3)OCC2)C5=CC=CC=N5
Molecular Formula
C24H23F4N5O3S
Molecular Weight
537.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Popular Products