MK-5046

CAT: 0931-MF-0095912-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0095912-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1022152-70-0
Target
Bombesin Receptor
Related Pathways
GPCR/G Protein
Purity
0.9991
Bioactivity
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM) .
Smiles
O[C@@](Cc1nc(CC2(CC2)C(F)(F)F)c[nH]1)(c1ccc(cc1)-n1cccn1)C(F)(F)F
Molecular Formula
C20H18F6N4O
Molecular Weight
444.37
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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