CDK4-IN-1

CAT:
931-T2082-01
Size:
25 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
CDK4-IN-1 - image 1

CDK4-IN-1

  • Target:

    CDK
  • Related Pathways:

    Cell Cycle/Checkpoint
  • Bioactivity:

    CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50=5.265 uM) respectively.
  • Smiles:

    CC(C)c1c(c(n[nH]1)Cl)c1nc(ncc1)Nc1ncc(cc1)N1CCC(CC1)N(C)C
  • Molecular Formula:

    C22H29ClN8
  • Molecular Weight:

    440.97
  • Shipping Conditions:

    Cool pack
  • Storage Temperature:

    -20°C
  • CAS Number:

    1256963-02-6