Products for Research Use Only
RegisterLogin

PROTAC ER Degrader-3

CAT: 0931-T18607-01Size: 100 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T18607-01Size:100 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
2158322-29-1
Target
Estrogen Receptor/ERR, PROTACs, Others
Related Pathways
Others, PROTAC, Endocrinology/Hormones
Bioactivity
PROTAC ER Degrader-3, an intermediate for the synthesis of PAC, specifically compound LP2. PAC serves as the linker for ADCs and PROTACs that are conjugated to an antibody. Notably, when PAC is conjugated to an antibody, it exhibits enhanced degradation of estrogen receptor-alpha (ERα) compared to PROTAC alone [1].
Smiles
CCC(=C(c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)c2ccc(cc2)C(=O)N2[C@@H](C)[C@H](NC(=O)[C@H](C)N(C)C(=O)OC(C)(C)C)C(=O)N(Cc3c(OC)ccc4ccccc34)c3ccc(cc23)C#N)cc1)c1ccccc1 |w:3.11|
Molecular Formula
C71H77N7O12
Molecular Weight
1220.434
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Related Products

CatalogName
T210250-01PROTAC ERα Degrader-9
T18605-01PROTAC ERα Degrader-2
T13839-01PROTAC ER Degrader-4
T208968-01PROTAC ER Degrader-12
T87264-01PROTAC ERα Degrader-7
T18606-01PROTAC ER Degrader-2
T210675-01PROTAC ERα Degrader-11
T204651-01PROTAC ER Degrader-15
T210833-01PROTAC ERα Degrader-12
T208971-01PROTAC ERα Degrader-6

Alternative Products

CatalogName
HY-175459PROTAC FAK degrader 3
HY-168551-01PROTAC ALK degrader-3
HY-135558PROTAC BRD4 Degrader-3
HY-161930PROTAC GPX4 degrader-3
HY-128527PROTAC ER Degrader-3
MBS5800292PROTAC IRAK4 degrader-3
MBS5820728PROTAC BTK Degrader-3
GTR19277025-01PROTAC HDAC8 Degrader-3
GTR19262351-01PROTAC STAT3 degrader-3
GTR19225039-01PROTAC FKBP Degrader-3

Popular Products