MK-4256

• Target :

  Others|||Somatostatin

• Related Pathways :

  Others|||GPCR/G Protein

• Bioactivity :

  MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively) .

• Smiles :

  Cc1nc(no1)[C@@]1(N[C@H](Cc2c1[nH]c1ccccc21)c1ncc([nH]1)-c1ccc(F)cc1)c1cnn(C)c1

• Molecular Formula :

  C27H23FN8O

• Molecular Weight :

  494.52

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1104599-69-0