MK-4256

• Target:

  Others|||Somatostatin

• Related Pathways:

  Others|||GPCR/G Protein

• Bioactivity:

  MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively) .

• Smiles:

  Cc1nc(no1)[C@@]1(N[C@H](Cc2c1[nH]c1ccccc21)c1ncc([nH]1)-c1ccc(F)cc1)c1cnn(C)c1

• Molecular Formula:

  C27H23FN8O

• Molecular Weight:

  494.52

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1104599-69-0