CJ-42794

• Target :

  Others|||Prostaglandin Receptor

• Related Pathways :

  GPCR/G Protein|||Immunology/Inflammation|||Others

• Purity :

  0.9992

• Bioactivity :

  CJ-42794 (CJ-042794) is a selective antagonist of the prostaglandin E receptor subtype 4 (EP4), inhibiting [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5. It exhibits a binding affinity that is at least 200-fold more selective for the human EP4 receptor than for other human EP receptor subtypes (EP1, EP2, and EP3) (IC50: 8.5 (pKi) ) .

• Smiles :

  C[C@H](NC(=O)c1cc(Cl)ccc1Oc1ccc(F)cc1)c1ccc(cc1)C(O)=O

• Molecular Formula :

  C22H17ClFNO4

• Molecular Weight :

  413.83

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  847728-01-2