MZP-54

• Target:

  Epigenetic Reader Domain|||PROTACs

• Related Pathways:

  PROTAC|||Chromatin/Epigenetic

• Bioactivity:

  MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology (Kd of 4 nM for Brd4BD2)

• Smiles:

  N ([C@H]1C=2C (N (C (C) =O) [C@@H] (C) C1) =CC=C (C2) C3=CC=C (C (NCCOCCOCCOCC (N[C@H] (C (=O) N4[C@H] (C (NCC5=CC=C (C=C5) C=6SC=NC6C) =O) C[C@@H] (O) C4) [C@@] (C) (C) C) =O) =O) C=C3) C7=CC=C (Cl) C=C7

• Molecular Formula:

  C55H66ClN7O9S

• Molecular Weight:

  1036.67

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2010159-47-2