MZP-55

• Target:

  Epigenetic Reader Domain|||PROTACs

• Related Pathways:

  Chromatin/Epigenetic|||PROTAC

• Bioactivity:

  MZP-55 is a selective BRD3/4 degrader based on PROTAC technology (Brd4BD2 with Kd of 8 nM)

• Smiles:

  N([C@H]1C=2C(N(C(C)=O)[C@@H](C)C1)=CC=C(C2)C3=CC=C(C(NCCOCCOCCOCCOCC(N[C@H](C(=O)N4[C@H](C(NCC5=CC=C(C=C5)C6=C(C)N=CS6)=O)C[C@@H](O)C4)[C@](C)(C)C)=O)=O)C=C3)C7=CC=C(Cl)C=C7

• Molecular Formula:

  C57H70ClN7O10S

• Molecular Weight:

  1080.73

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2010159-48-3