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GNE-0439

CAT: 0931-T11437-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-T11437-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1241902-40-8
Target
Sodium Channel
Related Pathways
Membrane transporter/Ion channel
Purity
0.996
Bioactivity
GNE-0439 is a novel, Nav1.7-selective inhibitor with an IC50 of 0.34 uM that also inhibits Nav1.5 (IC50=38.3 uM) and mutant N1742K channels (IC50=0.37 uM), possessing a carboxylic acid group that binds outside the channel pore, distinguishing it from known selective VSD4 binders and making it a valuable tool for ion channel research.
Smiles
C(N[C@@H]([C@@H](C)C)C(O)=O)(=O)C1=CC=C(C=C1)C2CCC(CCC)CC2
Molecular Formula
C21H31NO3
Molecular Weight
345.48
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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