Iloperidone-d3

CAT: 0804-HY-17410S-01Size: 100 mgDry Ice: NoHazardous: No
CAT#:0804-HY-17410S-01Size:100 mg
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Description
Iloperidone-d3 is the deuterium labeled Iloperidone. Iloperidone (HP 873) is a D2/5-HT2 receptor antagonist. Iloperidone is an atypical antipsychotic for the schizophrenia symptoms[1][2].
CAS Number
[1071167-49-1]
UNSPSC
12352005
Hazard Statement
H300
Target
5-HT Receptor; Dopamine Receptor; Isotope-Labeled Compounds
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Neuronal Signaling; Others
Field of Research
Neurological Disease
Solubility
10 mM in DMSO
Smiles
FC1=CC=C(C(C2CCN(CC2)CCCOC3=C(C=C(C=C3)C(C)=O)OC([2H])([2H])[2H])=NO4)C4=C1
Molecular Formula
C24H24D3FN2O4
Molecular Weight
429.50
Precautions
P264-P270-P330-P405-P501
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216. |[2]Kongsamut, S., et al., Iloperidone binding to human and rat dopamine and 5-HT receptors. Eur J Pharmacol, 1996. 317 (2-3) : p. 417-23.|[3]Sainati, S.M., et al., Safety, tolerability, and effect of food on the pharmacokinetics of iloperidone (HP 873), a potential atypical antipsychotic. J Clin Pharmacol, 1995. 35 (7) : p. 713-20.|[4]Albers, L.J., A. Musenga, and M.A. Raggi, Iloperidone: a new benzisoxazole atypical antipsychotic drug. Is it novel enough to impact the crowded atypical antipsychotic market? Expert Opin Investig Drugs, 2008. 17 (1) : p. 61-75.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Isoform
D3 Receptor

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Alternative Products

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164477Iloperidone-d3
163671Desfluoro Iloperidone-d3 (Impurity)
sc-499489Desfluoro iloperidone-d3 impurity
166179(R) -Hydroxy Iloperidone-d3
TRC-H943232-25MG(R)-Hydroxy Iloperidone-d3
sc-490759(S) -Hydroxy Iloperidone-d3
sc-488068Iloperidone Carboxylic Acid-d3
166438S-Hydroxy Iloperidone-d3
TRC-H943237-25MG(S)-Hydroxy Iloperidone-d3
MBS5753318Iloperidone metabolite Hydroxy Iloperidone

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