CB1R Allosteric modulator 3
CAT:
804-HY-150056-01
Size:
5 mg
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
CB1R Allosteric modulator 3
- CAS Number: 2633686-36-7
- UNSPSC Description: CB1R Allosteric modulator 3 is a CB1R positive allosteric modulator. CB1R Allosteric modulator 3 has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM, respectively[1].
- Target Antigen: Arrestin; Cannabinoid Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein;Neuronal Signaling
- Applications: Neuroscience-Neuromodulation
- Field of Research: Neurological Disease
- Assay Protocol: https://www.medchemexpress.com/cb1r-allosteric-modulator-3.html
- Solubility: DMSO : 100 mg/mL (ultrasonic)
- Smiles: ClC1=C(C=CC=C1)C(C2=C(C3=CC=CC=C3)NC4=C2C=CC=C4)C[N+]([O-])=O
- Molecular Weight: 376.84
- References & Citations: [1]Peter C Schaffer, et al. Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor agonist-positive allosteric modulator: site-III aromatic-ring congeners with enhanced activity and solubility. Bioorg Med Chem. 2020 Nov 1;28(21):115727.
- Shipping Conditions: Room Temperature
- Clinical Information: No Development Reported