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Prasugrel-13C6

CAT: 0804-HY-15284S3Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-15284S3Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Prasugrel-13C6 is a deuterated labeled Prasugrel[1]. Prasugrel (PCR 4099), a thienopyridine and proagent, inhibits platelet function. Prasugrel is an orally active and potent P2Y12 receptor antagonist, and inhibits ADP-induced platelet aggregation[2].
CAS Number
1261394-83-5
Product Name Alternative
PCR 4099-13C6
UNSPSC
12352005
Target
Isotope-Labeled Compounds; P2Y Receptor
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Others
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/prasugrel-13c6.html
Smiles
O=C(C1CC1)C([13C]2=[13C]([13CH]=[13CH][13CH]=[13CH]2)F)N3CC4=C(SC(OC(C)=O)=C4)CC3
Molecular Formula
C14 13C6H20FNO3S
Molecular Weight
379.40
References & Citations
[1]Wijeyeratne YD, et al. Anti-platelet therapy: ADP receptor antagonists. Br J Clin Pharmacol. 2011 Oct;72 (4) :647-57.|[2]Sugidachi A, et al. The greater in vivo antiplatelet effects of prasugrel as compared to clopidogrel reflect more efficient generation of its active metabolite with similar antiplatelet activity to that of clopidogrel's active metabolite. J Thromb Haemost. 2007 Jul;5 (7) :1545-51.|[3]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53 (2) :211-216.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported