Products for Research Use Only
RegisterLogin

Prasugrel-d5

CAT: 0804-HY-15284SSize: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-15284SSize:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Prasugrel-d5 is deuterium labeled Prasugrel. Prasugrel (PCR 4099), a thienopyridine and prodrug, inhibits platelet function. Prasugrel is an orally active and potent P2Y12 receptor antagonist, and inhibits ADP-induced platelet aggregation[1].
CAS Number
1127252-92-9
Product Name Alternative
PCR 4099-d5
UNSPSC
12352005
Target
Isotope-Labeled Compounds; P2Y Receptor
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Others
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Solubility
10 mM in DMSO
Smiles
FC1=CC=CC=C1C(N2CCC3=C(C=C(OC(C)=O)S3)C2)C(C4([2H])C([2H])([2H])C4([2H])[2H])=O
Molecular Formula
C20H15D5FNO3S
Molecular Weight
378.47
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216.|[2]Sugidachi A, et al. The greater in vivo antiplatelet effects of prasugrel as compared to clopidogrel reflect more efficient generation of its active metabolite with similar antiplatelet activity to that of clopidogrel's active metabolite. J Thromb Haemost. 2007 Jul;5 (7) :1545-51.|[3]Wijeyeratne YD, et al. Anti-platelet therapy: ADP receptor antagonists. Br J Clin Pharmacol. 2011 Oct;72 (4) :647-57.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Isoform
P2Y12 Receptor

Related Products

CatalogName
HY-15284-01Prasugrel
HY-15284S3Prasugrel-13C6
HY-15284S2-01Prasugrel-d4
HY-15284S1-01Prasugrel-d3
HY-15284A-01Prasugrel (hydrochloride)
HY-15284R-01Prasugrel (Standard)
HY-W704031Prasugrel metabolite 1
HY-W128916S-01Prasugrel metabolite-d4
HY-W686186-01Prasugrel hydroxy thiolactone
HY-15284BPrasugrel (Maleic acid)

Alternative Products

CatalogName
TRC-P701152-1MGPrasugrel-d5
TRC-P701167-5MGPrasugrel Thiolactone-d5 (Mixture of Diastereomers)
A1607-5Prasugrel

Popular Products