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Rel-Delequamine

CAT: 0804-HY-106874BSize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-106874BSize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Rel-Delequamine (rel-RS-15385-197) is an orally active, brain-penetrant, potent and selective M2-adrenoceptor antagonist and α2-adrenoceptor antagonist. rel-Delequamine has a pKi of 9.45 for α2-adrenoceptors in the rat cortex. rel-Delequamine augments K+-evoked release of noradrenaline with an EC50 of 1 nM[1].
CAS Number
119813-87-5
Product Name Alternative
Rel-RS-15385-197
UNSPSC
12352005
Target
Adrenergic Receptor; Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/rel-delequamine.html
Smiles
O=S(N1CCC[C@@]2(CN([C@]3(C[C@]12[H])[H])CCC4=C3C=CC(OC)=C4)[H])(C)=O
Molecular Formula
C18H26N2O3S
Molecular Weight
350.48
References & Citations
[1]Brown CM, et al. The pharmacology of RS-15385-197, a potent and selective alpha 2-adrenoceptor antagonist. Br J Pharmacol. 1993 Feb;108 (2) :516-25.|[2]Redfern WS, et al. Modulation of central noradrenergic function by RS-15385-197. Br J Pharmacol. 1993 Feb;108 (2) :526-33.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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