N-Desmethyl Eletriptan

N-Desmethyl Eletriptan

• CAS Number: 153525-55-4
• UNSPSC Description: N-desmethyl Eletriptan is a metabolite of Eletriptan (HY-A0039). It is formed from eletriptan primarily by the cytochrome P450 (CYP) isoform CYP3A4 in human liver microsomes.
• Target Antigen: Cytochrome P450
• Type: Reference compound
• Related Pathways: Metabolic Enzyme/Protease
• Applications: Metabolism-protein/nucleotide metabolism
• Field of Research: Metabolic Disease
• Assay Protocol: https://www.medchemexpress.com/n-desmethyl-eletriptan.html
• Smiles: O=[S](CCC1=CC=C2C(C(C[C@H]3CCCN3)=CN2)=C1)(C4=CC=CC=C4)=O
• Molecular Weight: 368.49
• References & Citations: [1]Evans, et al. Eletriptan metabolism by human hepatic CYP450 enzymes and transport by human P-glycoprotein. Drug Metab. Dispos. 31(7), 861-869 (2003).
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported