ERK2-IN-4

ERK2-IN-4

• CAS Number: 933786-58-4
• UNSPSC Description: ERK2-IN-4 (Compound 6o) is an effective and selective ERK2 inhibitor with a Ki of 0.006 μM. ERK2-IN-4 inhibits the ERK signaling pathway and can be used in cancer research[1].
• Target Antigen: ERK
• Type: Reference compound
• Related Pathways: MAPK/ERK Pathway;Stem Cell/Wnt
• Applications: Cancer-Kinase/protease
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/erk2-in-4.html
• Solubility: 10 mM in DMSO
• Smiles: OCC(C1=CC=C(C(Cl)=C1)F)NC(C2=CC(C(NN=C3)=C3C4=CC(Cl)=CC=C4)=CN2)=O
• Molecular Weight: 459.30
• References & Citations: [1]Aronov, Alex M et al. “Flipped out: structure-guided design of selective pyrazolylpyrrole ERK inhibitors.” Journal of medicinal chemistry vol. 50,6 (2007): 1280-7.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported