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Theliatinib

CAT: 0026-B3004-1Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0026-B3004-1Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Theliatinib is a potent epidermal growth factor receptor EGFR tyrosine kinase inhibitor with a Ki value of 0.05 nM and IC₅₀ of 3 nM. It exhibits strong antitumor activity in patient-derived estrogen cancer xenograft (PDECX) models with high EGFR expression, including remarkable tumor regression in two PDECX models with both EGFR gene amplification and protein overexpression in a dose-dependent manner (5 and 15 mg/kg/day). The efficacy of theliatinib is reduced in the models with PI3KCA mutations or FGFR1 overexpression in addition to high EGFR expression.
Shipping Conditions
RT
Storage Conditions
-20ºC
Shelf Life
36 months

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