Products for Research Use Only

Theliatinib (HMPL-309)

CAT: 0957-S8584Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-S8584Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Theliatinib (HMPL-309) is a highly potent EGFR inhibitor with Ki value of 0.05 nM against the wild type EGFR and IC50 values of 3 nM and 22 nM against EGFR and EGFR T790M/L858R mutant. It demonstrats 50 fold greater selectivity for EGFR compared to 72 other kinases.
CAS Number
1353644-70-8
Target
EGFR
Activity
Protein Tyrosine Kinase
Molecular Formula
C25H26N6O2
Storage Conditions
3 years -20°C powder