Succinate/succinate receptor antagonist 1
CAT:
804-HY-150205-03
Size:
25 mg
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

Succinate/succinate receptor antagonist 1
- CAS Number: 2361972-29-2
- UNSPSC Description: Succinate/succinate receptor antagonist 1 (compound 7a) is a succinate/succinate receptor antagonist. Succinate/succinate receptor antagonist 1 blocks succinate signaling in gingival tissue. Succinate/succinate receptor antagonist 1 inhibits the activation of succinate receptor 1 (SucnRl) with an IC50 value of 20 μΜ. Succinate/succinate receptor antagonist 1 can be used for the research of periodontal disease[1].
- Target Antigen: Others
- Type: Reference compound
- Related Pathways: Others
- Applications: COVID-19-immunoregulation
- Field of Research: Inflammation/Immunology
- Assay Protocol: https://www.medchemexpress.com/succinate-succinate-receptor-antagonist-1.html
- Solubility: DMSO : 25 mg/mL (ultrasonic)
- Smiles: O=C(NC)CC1=CC=C(C2=NC3=NC=CC=C3C=C2)C=C1
- Molecular Weight: 277.32
- References & Citations: [1]LI, Xin, et al. PERIODONTAL DISEASE THERAPY. WO2019136022. 2020.
- Shipping Conditions: Room Temperature
- Clinical Information: No Development Reported