L-803087

CAT: 0804-HY-108497-01Size: 1 mgDry Ice: NoHazardous: No

1 / 1

CAT#:0804-HY-108497-01Size:1 mg

Selected

24/48H Stock Items & 2 to 6 Weeks non Stock Items.

Quick Request Actions

Description

L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM. L-803087 is >280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice[1][2].

CAS Number

217480-26-7

UNSPSC

12352005

Target

Somatostatin Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Cancer-programmed cell death

Field of Research

Cancer; Neurological Disease

Assay Protocol

https://www.medchemexpress.com/l-803087.html

Purity

99.66

Solubility

DMSO : 250 mg/mL (ultrasonic)

Smiles

N=C(N)NCCC[C@@H](C(OC)=O)NC(CCCC1=C(C2=CC=CC=C2)NC3=C1C=C(F)C=C3F)=O

Molecular Formula

C25H29F2N5O3

Molecular Weight

485.53

References & Citations

[1]Rohrer SP, et al. Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry. Science. 1998 Oct 23;282 (5389) :737-40.|[2]Moneta D, et al. Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice. Eur J Neurosci. 2002 Sep;16 (5) :843-9.

Shipping Conditions

Blue Ice

Storage Conditions

-20°C, 3 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Related Products

Catalog	Name
HY-W928653	L-Seryl-L-leucyl-L-leucyl-L-lysine
HY-101552A-01	L, L-Dityrosine
HY-P4621-01	L-Alanyl-L-alanyl-L-glutamine
HY-W010789-01	L-Lysyl-L-tyrosine-α-L-lysine
HY-P4257	L-Isoleucyl-L-arginine
HY-129263-01	L-Isoleucyl-L-valine
HY-W101499-01	L-a-Aspartyl-L-leucine
HY-W101298-01	L-Leucyl-L-isoleucine
HY-W011607-01	L-Alanyl-L-tryptophan
HY-112171-01	γ-L-Glutamyl-L-alanine

Alternative Products

Catalog	Name
453095-01	L 803087
T11800-01	L-803087
T39207-01	L-803087 TFA
CCP1053-01	A-L-A-L
453309-01	L-Glycyl-L-lysyl-L-leucyl-L-isoleucyl-L-tyrosyl-L-seryl-L-alanyl-L-seryl-L-phenylalanyl-L-leucyl-L-tyrosyl-L-seryl-L-glycyl-L-valyl-L-prolyl-L-seryl-L-arganine
453434-01	L-Seryl-L-threonyl-L-glycyl-L-isoleucyl-L-seryl-L-valyl-L-prolyl-L-glycyl-L-prolyl-L-methionyl-L-glycyl-L-prolyl-L-seryl-L-glycyl-L-prolyl-L-Arginine
JH918176	L-Arginine, L-valyl-L-seryl-L-arginyl-L-arginyl-L-arginyl-L-arginyl-L-arginyl-L-arginylglycylglycyl-L-arginyl-L-arginyl-L-arginyl-
453216-01	L-Arginyl-L-valyl-L-α-aspartyl-L-prolyl-L-valyl-L-asparaginyl-L-phenylalanyl-L-lysyl-L-leucyl-L-leucyl-L-seryl-L-histidine
453308-01	L-Glycyl-L-arginyl-L-phenylalanyl-L-isoleucyl-L-threonyl-L-seryl-L-alanyl-L-aspartyl-L-threonyl-L-lysine
918629-48-8	L-Alanyl-L-Cysteinyl-L-Seryl-L-Seryl-L-Seryl-L-Prolyl-L-Seryl-L-Lysyl-L-Histidyl-L-Cysteinylglycine

L-803087

Related Products

Alternative Products

Popular Products