L-803087 TFA

• Target :

  Others|||Somatostatin

• Related Pathways :

  Others|||GPCR/G Protein

• Bioactivity :

  L-803087 TFA is a highly potent and selective agonist of the somatostatin sst4 receptor, exhibiting a Ki value of 0.7 nM. It displays a remarkable selectivity, being over 280-fold more preferential for the sst4 receptor compared to other somatostatin receptors. Furthermore, L-803087 TFA promotes AMPA-mediated synaptic responses in hippocampal preparations and enhances kainate-induced seizures in mice.

• Smiles :

  OC(=O)C(F)(F)F.COC(=O)[C@H](CCCNC(N)=N)NC(=O)CCCc1c([nH]c2c(F)cc(F)cc12)-c1ccccc1

• Molecular Formula :

  C27H30F5N5O5

• Molecular Weight :

  599.55

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1786412-46-1