L-803087

CAT:

931-T11800-01

Size:

1 mg

Price:

Ask

Target :
Somatostatin
Related Pathways :
GPCR/G Protein
Purity :
0.9937
Bioactivity :
L-803087 is a potent and selective agonist of the growth inhibitor sst4 receptor with a Ki value of 0.7 nM for sst4, demonstrating over 280-fold selectivity compared to other growth inhibitory receptors. L-803087 induces AMPA-mediated synaptic responses in the hippocampus in vitro and increases seizures in alginate-induced seizure-busting mice in vivo.
Smiles :
COC(=O)[C@H](CCCNC(N)=N)NC(=O)CCCc1c([nH]c2c(F)cc(F)cc12)-c1ccccc1
Molecular Formula :
C25H29F2N5O3
Molecular Weight :
485.53
Shipping Conditions :
Cool pack
Storage Temperature :
-20°C
CAS Number :
217480-26-7

Related Products

CAT	Name
T11800-01	L-803087
T39207-01	L-803087 TFA
T32812-01	L-Leucyl-L-prolyl-L-prolyl-L-seryl-L-arginine
T19396-01	L, L-Dityrosine
T22912-01	L-CCG-l
T19395-01	L, L-Dityrosine hydrochloride
T5593-01	L-Alanyl-L-glutamine
T9413-01	L-Alanyl-L-leucine
T34020	L-Phenylalanyl-L-leucine
T21053-01	L-Lysine L-glutamate

CAT	Name
574369	L-803087
M32990-01	L-803087
453095-01	L 803087
MBS5753384	L-803087
HY-108497-01	L-803087
BUP09477-01	L-803087
HY-108497A	L-803087 (TFA)
MBS5799730	L-803087 TFA
453309-01	L-Glycyl-L-lysyl-L-leucyl-L-isoleucyl-L-tyrosyl-L-seryl-L-alanyl-L-seryl-L-phenylalanyl-L-leucyl-L-tyrosyl-L-seryl-L-glycyl-L-valyl-L-prolyl-L-seryl-L-arganine
453434-01	L-Seryl-L-threonyl-L-glycyl-L-isoleucyl-L-seryl-L-valyl-L-prolyl-L-glycyl-L-prolyl-L-methionyl-L-glycyl-L-prolyl-L-seryl-L-glycyl-L-prolyl-L-Arginine