PAT-IN-1

• UNSPSC Description:

  PAT-IN-1 is a protein acyl transferases (PAT) inhibitor. PAT-IN-1 competitively inhibits Erf2 autopalmitoylation (WO2017011518A1; compound 13)[1].

• Target Antigen:

  Ras

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;MAPK/ERK Pathway

• Applications:

  Cancer-Kinase/protease

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/pat-in-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  CC(C1=CC=C(C=C1)CC(C)C)CN(CCN(C2)CCCC[C@@H]3N(CCNC3)CC(C4=CC=C(C=C4)CC(C)C)C)[C@H]2CC5=CC=C(C=C5)O

• Molecular Weight:

  681.05

• References & Citations:

  [1]Robert Joseph DESCHENES, et al. Protein acyl transferase inhibitors and methods of treatment. WO2017011518A1.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2066571-97-7