CYP1B1-IN-2

CYP1B1-IN-2

• CAS Number: 727730-24-7
• UNSPSC Description: CYP1B1-IN-2 (compound 9j) is a potent and selective CYP1B1 (cytochrome P450 1B1) inhibitor, with an IC50 of 0.52 nM[1].
• Target Antigen: Cytochrome P450
• Type: Reference compound
• Related Pathways: Metabolic Enzyme/Protease
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/cyp1b1-in-2.html
• Solubility: 10 mM in DMSO
• Smiles: O=C1C=C(C2=CC=CC(C(F)(F)F)=C2)OC3=C1C=CC4=CC=CC=C43
• Molecular Weight: 340.30
• References & Citations: [1]Dong J, et al. Synthesis and structure-activity relationship studies of α-naphthoflavone derivatives as CYP1B1 inhibitors. Eur J Med Chem. 2020 Feb 1;187:111938.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported