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CB1-IN-2

CAT: 0804-HY-147821Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-147821Size:1 Each
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CB1-IN-2 (Compound 4g) is a selective CB1 inhibitor with an IC50 of 0.644 μM. CB1-IN-2 can penetrates BBB and might cause CNS side effect similar with Rimonabant[1].
CAS Number
[2527805-39-4]
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/cb1-in-2.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=NN(C2=CC=C(Cl)C=C2Cl)C(C3CC3)=N1)NN4CCCCC4
Molecular Formula
C17H19Cl2N5O
Molecular Weight
380.27
References & Citations
[1]Tsai SE, et al. Chlorotrimethylsilane promoted one-flask heterocyclic synthesis of 1,2,4-triazoles from nitrilimines: Modeling studies and bioactivity evaluation of LH-21 and Rimonabant analogues. Bioorg Chem. 2020 Nov;104:104299.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB1

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