Rel-Ecopipam (hydrobromide)

• Description :

  Rel-Ecopipam (rel-SCH 39166) (Compound 6b) hydrobromide is a D1 receptor antagonist (Ki: 1.30 nM) [1].

• Product Name Alternative :

  Rel-SCH 39166 (hydrobromide)

• UNSPSC :

  12352005

• Target :

  Dopamine Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Neuronal Signaling

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Neurological Disease

• Assay Protocol :

  https://www.medchemexpress.com/rel-ecopipam-hydrobromide.html

• Solubility :

  10 mM in DMSO

• Smiles :

  CN1[C@]2([H])[C@@](C3=CC=CC=C3CC2)([H])C4=CC(O)=C(Cl)C=C4CC1.Br

• Molecular Formula :

  C19H21BrClNO

• Molecular Weight :

  394.73

• References & Citations :

  [1]Clark AH, et al. Assessment of dopamine D₁ receptor affinity and efficacy of three tetracyclic conformationally-restricted analogs of SKF38393. Bioorg Med Chem. 2011 Sep 15;19 (18) :5420-31.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• CAS Number :

  [1227675-51-5]