RyRs activator 1

RyRs activator 1

• CAS Number: 2571579-14-9
• UNSPSC Description: RyRs activator 1 (compound 7f) is a potent activator of ryanodine receptors (RyRs). RyRs activator 1 at 0.5 mg/L displays 100% larvicidal activity. The larvicidal activity of RyRs activator 1 is 90% at 0.01 mg/L[1].
• Target Antigen: Parasite
• Type: Reference compound
• Related Pathways: Anti-infection
• Applications: COVID-19-immunoregulation
• Field of Research: Infection
• Assay Protocol: https://www.medchemexpress.com/ryrs-activator-1.html
• Solubility: 10 mM in DMSO
• Smiles: O=C(C1=CC(C(F)(F)F)=NN1C2=CC([N+]([O-])=O)=CC=C2C#N)NC3=C(C(NC)=O)C=C(Cl)C=C3C
• Molecular Weight: 506.82
• References & Citations: [1] Liu J, et al. Discovery of a polysubstituted phenyl containing novel N-phenylpyrazole scaffold as potent ryanodine receptor activator. Bioorg Med Chem. 2020 Dec 15;28(24):115829
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported