ERK-IN-2

• Description:

  ERK-IN-2 is a ERK2 inhibitor with an IC50 value of 1.8 nM. ERK-IN-2 might lead to off-target toxicity and/or off-target activity at dose >10 μM[1].

• UNSPSC:

  12352005

• Target:

  ERK

• Type:

  Reference compound

• Related Pathways:

  MAPK/ERK Pathway; Stem Cell/Wnt

• Applications:

  Cancer-Kinase/protease

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/erk-in-2.html

• Solubility:

  10 mM in DMSO

• Smiles:

  OCC1=NC(NC(N[C@H](C)C2=CC=CC=C2)=O)=CC3=C1C=NN3.[H]Cl

• Molecular Formula:

  C16H18ClN5O2

• Molecular Weight:

  347.80

• References & Citations:

  [1]MRK-ERK Inhibitor and Negative Control

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• Isoform:

  ERK2

• CAS Number:

  [2743576-56-7]