GRK6-IN-3

• Description:

  GRK6-IN-3 is a G protein coupled receptor 6 kinase (GRK6) inhibitor with an IC50 1.03 μM[1].

• UNSPSC:

  12352005

• Hazard Statement:

  H315-H319-H320

• Target:

  G Protein-coupled Receptor Kinase (GRK)

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  COVID-19-immunoregulation

• Field of Research:

  Inflammation/Immunology

• Assay Protocol:

  https://www.medchemexpress.com/grk6-in-3.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(C1=C(N)N(CCCCC)C2=NC3=CC=CC=C3N=C21)OC

• Molecular Formula:

  C17H20N4O2

• Molecular Weight:

  312.37

• Precautions:

  P264-P280-P302+P352-P305+P351+P338-P362

• References & Citations:

  [1]Alexander Keith Stewart, et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458A2.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  499231-87-7