GRK6-IN-4

• Description:

  GRK6-IN-4 is a G protein coupled receptor 6 kinase (GRK6) inhibitor with an IC50 of 1.56 μM. GRK6-IN-4 can be utilized in research related to hematological malignancies, inflammatory diseases, and autoimmune disorders[1].

• UNSPSC:

  12352005

• Hazard Statement:

  H315-H319-H320

• Target:

  G Protein-coupled Receptor Kinase (GRK)

• Related Pathways:

  GPCR/G Protein

• Field of Research:

  Cancer; Inflammation/Immunology

• Smiles:

  N#CC1=C(N)N(CCCC)C2=C1N=C3C=CC=CC3=N2

• Molecular Formula:

  C15H15N5

• Molecular Weight:

  265.31

• Precautions:

  P264-P280-P302+P352-P305+P351+P338-P362

• References & Citations:

  [1]Alexander K.S., et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458A2. 2013-05-02

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  Phase 1

• CAS Number:

  300731-73-1