GRK6-IN-5

• Description :

  GRK6-IN-5 is a GRK6 polypeptide inhibitor, with IC50 value of 4.48 μΜ. GRK6-IN-5 can be used to study hematological malignancies, inflammation diseases, and autoimmune disorders[1].

• CAS Number :

  [33495-39-5]

• UNSPSC :

  12352005

• Target :

  G Protein-coupled Receptor Kinase (GRK)

• Related Pathways :

  GPCR/G Protein

• Field of Research :

  Cancer; Inflammation/Immunology

• Smiles :

  OC1=C(C(C2=NC=CC=C2)NC3=CC=C(C=C3)OCC)C=CC4=CC=CN=C14

• Molecular Formula :

  C23H21N3O2

• Molecular Weight :

  371.43

• References & Citations :

  [1]Alexander Keith Stewart, et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458. WIPO. 2012-10-26.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported