GRK6-IN-5

• Description:

  GRK6-IN-5 is a GRK6 polypeptide inhibitor, with IC50 value of 4.48 μΜ. GRK6-IN-5 can be used to study hematological malignancies, inflammation diseases, and autoimmune disorders[1].

• UNSPSC:

  12352005

• Target:

  G Protein-coupled Receptor Kinase (GRK)

• Related Pathways:

  GPCR/G Protein

• Field of Research:

  Cancer; Inflammation/Immunology

• Smiles:

  OC1=C(C(C2=NC=CC=C2)NC3=CC=C(C=C3)OCC)C=CC4=CC=CN=C14

• Molecular Formula:

  C23H21N3O2

• Molecular Weight:

  371.43

• References & Citations:

  [1]Alexander Keith Stewart, et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458. WIPO. 2012-10-26.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  33495-39-5