RS-5773

• Description :

  RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction [1].

• CAS Number :

  [129173-57-5]

• UNSPSC :

  12352005

• Target :

  Calcium Channel

• Type :

  Reference compound

• Related Pathways :

  Membrane Transporter/Ion Channel; Neuronal Signaling

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Neurological Disease; Cardiovascular Disease

• Assay Protocol :

  https://www.medchemexpress.com/rs-5773.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=C1[C@@H]([C@@H](SC2=CC(CC3=CC=CS3)=CC=C2N1CCN(C)C)C4=CC=C(C=C4)OC)OC(C)=O.[H]Cl

• Molecular Formula :

  C27H31ClN2O4S2

• Molecular Weight :

  547.13

• References & Citations :

  [1]H Shiga, et al. Antianginal effect of RS-5773, a diltiazem congener, in the methacholine-induced anginal model in rats. Jpn J Pharmacol . 1996 Dec;72 (4) :365-74.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported