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Asenapine (citrate)

CAT: 0804-HY-10121BSize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-10121BSize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Asenapine citrate, an atypical antipsychotic, is an antagonist of serotonin receptors (pKi: 8.4-10.5), adrenoceptors (pKi: 8.9-9.5), dopamine receptors (pKi: 8.9-9.4) and histamine receptors (pKi: 8.2-9.0) . Asenapine citrate can be used in the research of schizophrenia and bipolar disorder[1][2].
CAS Number
1411867-74-7
Product Name Alternative
Org 5222 (citrate)
UNSPSC
12352005
Target
5-HT Receptor; Adrenergic Receptor; Dopamine Receptor; Histamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/asenapine-citrate.html
Solubility
10 mM in DMSO
Smiles
ClC1=CC=C2OC3=CC=CC=C3[C@@](C4)([H])[C@](CN4C)([H])C2=C1.O=C(CC(C(O)=O)(O)CC(O)=O)O
Molecular Formula
C23H24ClNO8
Molecular Weight
477.89
References & Citations
[1]M Shahid, et al. Asenapine: a novel psychopharmacologic agent with a unique human receptor signature. J Psychopharmacol. 2009 Jan;23 (1) :65-73.|[2]Olivia Frånberg, et al. Asenapine, a novel psychopharmacologic agent: preclinical evidence for clinical effects in schizophrenia. Psychopharmacology (Berl) . 2008 Feb;196 (3) :417-29.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Launched
Isoform
D1 Receptor; D2 Receptor; D3 Receptor; D4 Receptor; H1 Receptor; H2 Receptor; mLAG-3; MUC2; MUC3; Prostaglandin D Synthase; α adrenergic receptor; α-1 microglobulin

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