K-(D-1-Nal)-FwLL-NH2 (TFA)

K-(D-1-Nal)-FwLL-NH2 (TFA)

• UNSPSC Description: K-(D-1-Nal)-FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
• Target Antigen: GHSR
• Type: Peptides
• Related Pathways: GPCR/G Protein
• Applications: Neuroscience-Neuromodulation
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/k-d-1-nal-fwll-nh2-tfa.html
• Solubility: 10 mM in DMSO
• Smiles: CC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=C5C=CC=CC5=CC=C4)NC([C@H](CCCCN)N)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F
• Molecular Weight: 1016.16
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported