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(±) -Penbutolol

CAT: 0804-HY-116790B-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-116790B-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
(±) -Penbutolol ((Rac) -Penbutolol) is the racemic mixture of Penbutolol. (±) -Penbutolol is an orally active β-adrenergic receptor antagonist. (±) -Penbutolol antagonizes exercise-induced tachycardia, reduces the increase in peak expiratory flow rate (PEFR) caused by exercise, and decreases resting plasma renin activity (PRA) . (±) -Penbutolol reaches peak plasma concentration 1 hour after oral administration, with a half-life of 4.5 hours, and is converted into an active metabolite in the body. (±) -Penbutolol can be used in cardiovascular-related disease research[1].
CAS Number
36507-48-9
Product Name Alternative
(Rac) -Penbutolol; (±) -Isopenbutolol
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/racemic-penbutolol.html
Smiles
OC(CNC(C)(C)C)COC1=CC=CC=C1C2CCCC2
Molecular Formula
C18H29NO2
Molecular Weight
291.43
References & Citations
[1]Giudicelli JF, et al. Comparative beta-adrenoceptor blocking effects and pharmacokinetics of penbutolol and propranolol in man. Br J Clin Pharmacol. 1977 Apr;4 (2) :135-40.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
β adrenergic receptor

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