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(±) -Penbutolol

CAT: 0931-T201472-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T201472-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
36507-48-9
Target
Adrenergic Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
(±) -Penbutolol ((Rac) -Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±) -Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.
Smiles
OC(COC=1C=CC=CC1C2CCCC2)CNC(C)(C)C
Molecular Formula
C18H29NO2
Molecular Weight
291.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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