P-CAB agent 2 (hydrochloride)

P-CAB agent 2 (hydrochloride)

• CAS Number: 2209911-80-6
• UNSPSC Description: P-CAB agent 2 hydrochloride is a potent and orally active potassium-competitive acid blocker and a gastric acid secretion inhibitor. P-CAB agent 2 hydrochloride inhibits H+/K+-ATPase activity with an IC50 value of IC50 value of 18.69 M. P-CAB agent 2 hydrochloride shows no acute toxicity and inhibits histamine (HY-B1204)-induced gastric acid secretion[1].
• Target Antigen: Potassium Channel
• Type: Reference compound
• Related Pathways: Membrane Transporter/Ion Channel
• Applications: Metabolism-protein/nucleotide metabolism
• Field of Research: Endocrinology
• Assay Protocol: https://www.medchemexpress.com/p-cab-agent-2-hydrochloride.html
• Solubility: DMSO : 100 mg/mL (ultrasonic)
• Smiles: O=S(C1=CC(OCCCOC)=CC=C1)(N2C=C(CNC)C=C2C3=C(F)C=CC=C3)=O.Cl
• Molecular Weight: 468.97
• References & Citations: [1]YinLin Qin, et al. Pyrrole sulfonyl derivative, and preparation method and medical use thereof. WO2016119505A1.
• Shipping Conditions: Room Temperature
• Clinical Information: No Development Reported